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Moreau_Deltamethrin

Notes


Deltamethrin PBK - Moreau et al. 2025 Stomach -> Duodenum -> GITissue -> Liver Perfusion-limited: Blood <-> Liver, Blood <-> Rest Hepatic metabolism: intrinsic clearance Plasma metabolism: set to 0 for BAP

Overview

key value
Modelled species/orgamism(s) not specified
Model chemical(s) not specified
Input route(s) no routes detected
Time resolution not specified
Amounts unit not specified
Volume unit not specified
Number of compartments 7
Number of species 9
Number of parameters 37 (20 external / 17 internal)

Diagram

Diagram

Compartments

id name unit model qualifier
Stomach not specified not specified not specified
GITissue not specified not specified not specified
Duodenum not specified not specified not specified
Liver not specified not specified not specified
Plasma not specified not specified not specified
Rest not specified not specified not specified
Urine not specified not specified not specified

Species

id name unit model qualifier
ASt not specified not specified not specified
ADuodenum not specified not specified not specified
AGITissue not specified not specified not specified
ALiver not specified not specified not specified
APlasma not specified not specified not specified
ARest not specified not specified not specified
ALiverMet not specified not specified not specified
APlasmaMet not specified not specified not specified
AUrine not specified not specified not specified

Transfer equations

id from to equation
_J0 ASt ADuodenum ksto * ASt
_J1 ADuodenum AGITissue kabs * ADuodenum
_J2 AGITissue ALiver QGI * CGITissue / PGI
_J3 APlasma AGITissue QGI * CPlasma
_J4 APlasma ALiver QL * CPlasma
_J5 ALiver APlasma (QL + QGI) * CLiver / PL
_J6 APlasma ARest QRest * CPlasma
_J7 ARest APlasma QRest * CRest / PRest
_J8 APlasma APlasmaMet CLintB * CPlasma
_J9 APlasma AUrine CLU * APlasma
_J10 ALiver ALiverMet CLintL * (CLiver / PL)

ODEs

\(\frac{d[\mathtt{ASt}]}{dt} = - \mathit{ksto}\cdot \mathit{ASt}\)

\(\frac{d[\mathtt{ADuodenum}]}{dt} = \mathit{ksto}\cdot \mathit{ASt} - \mathit{kabs}\cdot \mathit{ADuodenum}\)

\(\frac{d[\mathtt{AGITissue}]}{dt} = \mathit{kabs}\cdot \mathit{ADuodenum} - \frac{\mathit{QGI}\cdot \mathit{CGITissue}}{\mathit{PGI}} + \mathit{QGI}\cdot \mathit{CPlasma}\)

\(\frac{d[\mathtt{ALiver}]}{dt} = \frac{\mathit{QGI}\cdot \mathit{CGITissue}}{\mathit{PGI}} + \mathit{QL}\cdot \mathit{CPlasma} - \frac{(\mathit{QL}+\mathit{QGI})\cdot \mathit{CLiver}}{\mathit{PL}} - \mathit{CLintL}\cdot \frac{\mathit{CLiver}}{\mathit{PL}}\)

\(\frac{d[\mathtt{APlasma}]}{dt} = - \mathit{QGI}\cdot \mathit{CPlasma} - \mathit{QL}\cdot \mathit{CPlasma} + \frac{(\mathit{QL}+\mathit{QGI})\cdot \mathit{CLiver}}{\mathit{PL}} - \mathit{QRest}\cdot \mathit{CPlasma} + \frac{\mathit{QRest}\cdot \mathit{CRest}}{\mathit{PRest}} - \mathit{CLintB}\cdot \mathit{CPlasma} - \mathit{CLU}\cdot \mathit{APlasma}\)

\(\frac{d[\mathtt{ARest}]}{dt} = \mathit{QRest}\cdot \mathit{CPlasma} - \frac{\mathit{QRest}\cdot \mathit{CRest}}{\mathit{PRest}}\)

\(\frac{d[\mathtt{ALiverMet}]}{dt} = \mathit{CLintL}\cdot \frac{\mathit{CLiver}}{\mathit{PL}}\)

\(\frac{d[\mathtt{APlasmaMet}]}{dt} = \mathit{CLintB}\cdot \mathit{CPlasma}\)

\(\frac{d[\mathtt{AUrine}]}{dt} = \mathit{CLU}\cdot \mathit{APlasma}\)

Assignment rules

variable assignment
VL VLC * BW
VGITissue VGITissueC * BW
VUrine VUrineC * BW / 24 / 1000
VRest 0.84 * BW - VL - VGITissue - VPlasma
QCPlasma QC * (1 - Hct)
QGI QGIc * QC
QL QLc * QC
QRest QCPlasma - QL - QGI
CLintL CLintLC * VL
CLUC GFR
CLU Free * GFR
CGITissue AGITissue / GITissue
CLiver ALiver / Liver
CPlasma APlasma / Plasma
CRest ARest / Rest
CUrine AUrine / Urine
Met CLintL * (CLiver / PL)

Initial assignments

variable assignment
GITissue VGITissue
Liver VL
Plasma VPlasma
Rest VRest
Urine VUrine

Parameters

id name unit model qualifier
MW not specified not specified not specified
BW not specified not specified not specified
VLC not specified not specified not specified
VGITissueC not specified not specified not specified
VL not specified not specified not specified
VGITissue not specified not specified not specified
VPlasma not specified not specified not specified
VUrineC not specified not specified not specified
VUrine not specified not specified not specified
VRest not specified not specified not specified
QC not specified not specified not specified
Hct not specified not specified not specified
QCPlasma not specified not specified not specified
QGIc not specified not specified not specified
QLc not specified not specified not specified
QGI not specified not specified not specified
QL not specified not specified not specified
QRest not specified not specified not specified
PL not specified not specified not specified
PGI not specified not specified not specified
PRest not specified not specified not specified
ksto not specified not specified not specified
kabs not specified not specified not specified
Fa not specified not specified not specified
CLintLC not specified not specified not specified
CLintL not specified not specified not specified
CLintB not specified not specified not specified
Free not specified not specified not specified
GFR not specified not specified not specified
CLUC not specified not specified not specified
CLU not specified not specified not specified
CGITissue not specified not specified not specified
CLiver not specified not specified not specified
CPlasma not specified not specified not specified
CRest not specified not specified not specified
CUrine not specified not specified not specified
Met not specified not specified not specified