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OFlaherty 2001

Notes


Cr PBK (O'Flaherty et al. 2001):

Overview

key value
Modelled species/orgamism(s) http://purl.obolibrary.org/obo/NCBITaxon_9606
Model chemical(s) http://purl.obolibrary.org/obo/CHEBI_155866
Input route(s) 1 (oral)
Time resolution d
Amounts unit mg
Volume unit L
Number of compartments 6
Number of species 12
Number of parameters 30 (14 external / 16 internal)

Diagram

Diagram

Compartments

id name unit model qualifier
GI Gut compartment L http://purl.obolibrary.org/obo/PBPKO_00477
Liver Liver compartment L http://purl.obolibrary.org/obo/PBPKO_00558
Plasma Plasma compartment L http://purl.obolibrary.org/obo/PBPKO_00488
RBC Red blood cells compartment L http://purl.obolibrary.org/obo/PBPKO_00634
Rest Rest of body compartment L http://purl.obolibrary.org/obo/PBPKO_00450
Feces Feces compartment L http://purl.obolibrary.org/obo/PBPKO_00555

Species

id name unit model qualifier
AGI_Cr3 Amount in gut mg http://purl.obolibrary.org/obo/PBPKO_00496
AGI_Cr6 Amount in gut mg http://purl.obolibrary.org/obo/PBPKO_00496
ALiver_Cr3 Amount in liver mg http://purl.obolibrary.org/obo/PBPKO_00497
ALiver_Cr6 Amount in liver mg http://purl.obolibrary.org/obo/PBPKO_00497
Aplasma_Cr3 Amount in plasma mg http://purl.obolibrary.org/obo/PBPKO_00502
Aplasma_Cr6 Amount in plasma mg http://purl.obolibrary.org/obo/PBPKO_00502
ARBC_Cr3 Amount in red blood cells mg http://purl.obolibrary.org/obo/PBPKO_00623
ARBC_Cr6 Amount in red blood cells mg http://purl.obolibrary.org/obo/PBPKO_00623
ARest_Cr3 Amount in rest of body mg http://purl.obolibrary.org/obo/PBPKO_00501
ARest_Cr6 Amount in rest of body mg http://purl.obolibrary.org/obo/PBPKO_00501
AFeces_Cr3 Amount in feces mg http://purl.obolibrary.org/obo/PBPKO_00273
AFeces_Cr6 Amount in feces mg http://purl.obolibrary.org/obo/PBPKO_00273

Transfer equations

id from to equation
_J0 AGI_Cr6 AGI_Cr3 kred_GI * AGI_Cr6
_J1 AGI_Cr6 ALiver_Cr6 AGI_Cr6 * kabs_Cr6
_J2 AGI_Cr3 ALiver_Cr3 AGI_Cr3 * kabs_Cr3
_J3 AGI_Cr6 AFeces_Cr6 kfe * AGI_Cr6
_J4 AGI_Cr3 AFeces_Cr3 kfe * AGI_Cr3
_J5 ALiver_Cr6 ALiver_Cr3 kred_Liver * ALiver_Cr6
_J6 ALiver_Cr6 Aplasma_Cr6 kt_Plasma_Cr6 * ALiver_Cr6 / VL
_J7 ALiver_Cr3 Aplasma_Cr3 kt_Plasma_Cr3 * ALiver_Cr3 / VL
_J8 Aplasma_Cr6 Aplasma_Cr3 kred_Plasma * Aplasma_Cr6
_J9 Aplasma_Cr6 ALiver_Cr6 kt_Tissues_Cr6 * Aplasma_Cr6 / Vplasma
_J10 Aplasma_Cr3 ALiver_Cr3 kt_Tissues_Cr3 * Aplasma_Cr3 / Vplasma
_J11 ARBC_Cr6 ARBC_Cr3 kred_RBC * ARBC_Cr6
_J12 Aplasma_Cr6 ARBC_Cr6 kt_Tissues_Cr6 * Aplasma_Cr6 / Vplasma
_J13 Aplasma_Cr3 ARBC_Cr3 kt_Tissues_Cr3 * Aplasma_Cr3 / Vplasma
_J14 ARBC_Cr3 Aplasma_Cr3 kt_Plasma_Cr3 * ARBC_Cr3 / VRBC
_J15 ARBC_Cr6 Aplasma_Cr6 kt_Plasma_Cr6 * ARBC_Cr6 / VRBC
_J16 ARest_Cr6 Aplasma_Cr6 kt_Plasma_Cr6 * ARest_Cr6 / VRest
_J17 ARest_Cr3 Aplasma_Cr3 kt_Plasma_Cr3 * ARest_Cr3 / VRest
_J18 Aplasma_Cr6 ARest_Cr6 kt_Tissues_Cr6 * Aplasma_Cr6 / Vplasma
_J19 Aplasma_Cr3 ARest_Cr3 kt_Tissues_Cr3 * Aplasma_Cr3 / Vplasma

ODEs

\(\frac{d[\mathtt{AGI-Cr3}]}{dt} = \mathit{kred_{GI}}\cdot \mathit{AGI_{Cr6}} - \mathit{AGI_{Cr3}}\cdot \mathit{kabs_{Cr3}} - \mathit{kfe}\cdot \mathit{AGI_{Cr3}}\)

\(\frac{d[\mathtt{AGI-Cr6}]}{dt} = - \mathit{kred_{GI}}\cdot \mathit{AGI_{Cr6}} - \mathit{AGI_{Cr6}}\cdot \mathit{kabs_{Cr6}} - \mathit{kfe}\cdot \mathit{AGI_{Cr6}}\)

\(\frac{d[\mathtt{ALiver-Cr3}]}{dt} = \mathit{AGI_{Cr3}}\cdot \mathit{kabs_{Cr3}} + \mathit{kred_{Liver}}\cdot \mathit{ALiver_{Cr6}} - \frac{\mathit{kt\_Plasma\_Cr3}\cdot \mathit{ALiver_{Cr3}}}{\mathit{VL}} + \frac{\mathit{kt\_Tissues\_Cr3}\cdot \mathit{Aplasma_{Cr3}}}{\mathit{Vplasma}}\)

\(\frac{d[\mathtt{ALiver-Cr6}]}{dt} = \mathit{AGI_{Cr6}}\cdot \mathit{kabs_{Cr6}} - \mathit{kred_{Liver}}\cdot \mathit{ALiver_{Cr6}} - \frac{\mathit{kt\_Plasma\_Cr6}\cdot \mathit{ALiver_{Cr6}}}{\mathit{VL}} + \frac{\mathit{kt\_Tissues\_Cr6}\cdot \mathit{Aplasma_{Cr6}}}{\mathit{Vplasma}}\)

\(\frac{d[\mathtt{Aplasma-Cr3}]}{dt} = \frac{\mathit{kt\_Plasma\_Cr3}\cdot \mathit{ALiver_{Cr3}}}{\mathit{VL}} + \mathit{kred_{Plasma}}\cdot \mathit{Aplasma_{Cr6}} - \frac{\mathit{kt\_Tissues\_Cr3}\cdot \mathit{Aplasma_{Cr3}}}{\mathit{Vplasma}} - \frac{\mathit{kt\_Tissues\_Cr3}\cdot \mathit{Aplasma_{Cr3}}}{\mathit{Vplasma}} + \frac{\mathit{kt\_Plasma\_Cr3}\cdot \mathit{ARBC_{Cr3}}}{\mathit{VRBC}} + \frac{\mathit{kt\_Plasma\_Cr3}\cdot \mathit{ARest_{Cr3}}}{\mathit{VRest}} - \frac{\mathit{kt\_Tissues\_Cr3}\cdot \mathit{Aplasma_{Cr3}}}{\mathit{Vplasma}}\)

\(\frac{d[\mathtt{Aplasma-Cr6}]}{dt} = \frac{\mathit{kt\_Plasma\_Cr6}\cdot \mathit{ALiver_{Cr6}}}{\mathit{VL}} - \mathit{kred_{Plasma}}\cdot \mathit{Aplasma_{Cr6}} - \frac{\mathit{kt\_Tissues\_Cr6}\cdot \mathit{Aplasma_{Cr6}}}{\mathit{Vplasma}} - \frac{\mathit{kt\_Tissues\_Cr6}\cdot \mathit{Aplasma_{Cr6}}}{\mathit{Vplasma}} + \frac{\mathit{kt\_Plasma\_Cr6}\cdot \mathit{ARBC_{Cr6}}}{\mathit{VRBC}} + \frac{\mathit{kt\_Plasma\_Cr6}\cdot \mathit{ARest_{Cr6}}}{\mathit{VRest}} - \frac{\mathit{kt\_Tissues\_Cr6}\cdot \mathit{Aplasma_{Cr6}}}{\mathit{Vplasma}}\)

\(\frac{d[\mathtt{ARBC-Cr3}]}{dt} = \mathit{kred_{RBC}}\cdot \mathit{ARBC_{Cr6}} + \frac{\mathit{kt\_Tissues\_Cr3}\cdot \mathit{Aplasma_{Cr3}}}{\mathit{Vplasma}} - \frac{\mathit{kt\_Plasma\_Cr3}\cdot \mathit{ARBC_{Cr3}}}{\mathit{VRBC}}\)

\(\frac{d[\mathtt{ARBC-Cr6}]}{dt} = - \mathit{kred_{RBC}}\cdot \mathit{ARBC_{Cr6}} + \frac{\mathit{kt\_Tissues\_Cr6}\cdot \mathit{Aplasma_{Cr6}}}{\mathit{Vplasma}} - \frac{\mathit{kt\_Plasma\_Cr6}\cdot \mathit{ARBC_{Cr6}}}{\mathit{VRBC}}\)

\(\frac{d[\mathtt{ARest-Cr3}]}{dt} = - \frac{\mathit{kt\_Plasma\_Cr3}\cdot \mathit{ARest_{Cr3}}}{\mathit{VRest}} + \frac{\mathit{kt\_Tissues\_Cr3}\cdot \mathit{Aplasma_{Cr3}}}{\mathit{Vplasma}}\)

\(\frac{d[\mathtt{ARest-Cr6}]}{dt} = - \frac{\mathit{kt\_Plasma\_Cr6}\cdot \mathit{ARest_{Cr6}}}{\mathit{VRest}} + \frac{\mathit{kt\_Tissues\_Cr6}\cdot \mathit{Aplasma_{Cr6}}}{\mathit{Vplasma}}\)

\(\frac{d[\mathtt{AFeces-Cr3}]}{dt} = \mathit{kfe}\cdot \mathit{AGI_{Cr3}}\)

\(\frac{d[\mathtt{AFeces-Cr6}]}{dt} = \mathit{kfe}\cdot \mathit{AGI_{Cr6}}\)

Assignment rules

variable assignment
VL VLc * BW
Vplasma 0.55 * VRBC / 0.45
VRBC VRBCc * BW
VRest BW - VL - VRBC - Vplasma
CGI_Cr3 AGI_Cr3 / GI
CGI_Cr6 AGI_Cr6 / GI
CLiver_Cr3 ALiver_Cr3 / Liver
CLiver_Cr6 ALiver_Cr6 / Liver
CPlasma_Cr3 Aplasma_Cr3 / Plasma
CPlasma_Cr6 Aplasma_Cr6 / Plasma
CRBC_Cr3 ARBC_Cr3 / RBC
CRBC_Cr6 ARBC_Cr6 / RBC
CRest_Cr3 ARest_Cr3 / Rest
CRest_Cr6 ARest_Cr6 / Rest
CFeces_Cr3 AFeces_Cr3 / Feces
CFeces_Cr6 AFeces_Cr6 / Feces

Initial assignments

variable assignment
Liver VL
Plasma Vplasma
RBC VRBC
Rest VRest

Parameters

id name unit model qualifier
VL Volume of liver L http://purl.obolibrary.org/obo/PBPKO_00077
Vplasma Volume of plasma L http://purl.obolibrary.org/obo/PBPKO_00103
VRBC Volume of red blood cells L http://purl.obolibrary.org/obo/PBPKO_00108
VRest Volume of rest of body L http://purl.obolibrary.org/obo/PBPKO_00105
BW Bodyweight kg http://purl.obolibrary.org/obo/PBPKO_00008
VLc Volume fraction of liver dimensionless http://purl.obolibrary.org/obo/PBPKO_00078
VRBCc Volume fraction of red blood cells dimensionless not specified
CGI_Cr3 Concentration in gut mg/L http://purl.obolibrary.org/obo/PBPKO_00538
CGI_Cr6 Concentration in gut mg/L http://purl.obolibrary.org/obo/PBPKO_00538
CLiver_Cr3 Concentration in liver mg/L http://purl.obolibrary.org/obo/PBPKO_00539
CLiver_Cr6 Concentration in liver mg/L http://purl.obolibrary.org/obo/PBPKO_00539
CPlasma_Cr3 Concentration in plasma mg/L http://purl.obolibrary.org/obo/PBPKO_00549
CPlasma_Cr6 Concentration in plasma mg/L http://purl.obolibrary.org/obo/PBPKO_00549
CRBC_Cr3 Concentration in red blood cells mg/L http://purl.obolibrary.org/obo/PBPKO_00301
CRBC_Cr6 Concentration in red blood cells mg/L http://purl.obolibrary.org/obo/PBPKO_00301
CRest_Cr3 Concentration in rest of body mg/L http://purl.obolibrary.org/obo/PBPKO_00548
CRest_Cr6 Concentration in rest of body mg/L http://purl.obolibrary.org/obo/PBPKO_00548
CFeces_Cr3 Concentration in feces mg/L not specified
CFeces_Cr6 Concentration in feces mg/L not specified
kabs_Cr6 Rate constant for absorption of Cr(VI) from the GI tract mg/d http://purl.obolibrary.org/obo/PBPKO_00141
kabs_Cr3 Rate constant for absorption of Cr(III) from the GI tract mg/d http://purl.obolibrary.org/obo/PBPKO_00141
kt_Plasma_Cr6 Clearance of diffusible Cr(VI) from all other tissues into plasma (L/da) L/d not specified
kt_Plasma_Cr3 Clearance of diffusible Cr(III) from all other tissues into plasma (L/da) L/d not specified
kt_Tissues_Cr6 Clearance of diffusible Cr(VI) from plasma into all tissues (L/da) L/d not specified
kt_Tissues_Cr3 Clearance of diffusible Cr(III) from plasma into all tissues (L/da) L/d not specified
kred_GI Rate constant for reduction of Cr(VI) to Cr(III) in GI mg/d not specified
kred_Liver Rate constant for reduction of Cr(VI) to Cr(III) in GI mg/d not specified
kred_RBC Rate constant for reduction of Cr(VI) to Cr(III) in plasma mg/d not specified
kred_Plasma Rate constant of reduction in plasma mg/d not specified
kfe First-order rate constant for passage of Cr out of the absorption region of the GI tract /d not specified