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ElMasri 2008

Notes


Arsene ElMasri et al. 2008

Overview

key value
Modelled species/orgamism(s) http://purl.obolibrary.org/obo/NCBITaxon_9606
Model chemical(s) http://purl.obolibrary.org/obo/CHEBI_190436
Input route(s) 2 (oral, inhalation)
Time resolution h
Amounts unit mol
Volume unit dimensionless
Number of compartments 8
Number of species 32
Number of parameters 78 (33 external / 45 internal)

Diagram

Diagram

Compartments

id name unit model qualifier
Lumen Compartment of lumen dimensionless http://purl.obolibrary.org/obo/PBPKO_00478
Gut Compartment of Gut dimensionless http://purl.obolibrary.org/obo/PBPKO_00477
Liver Compartment of liver dimensionless http://purl.obolibrary.org/obo/PBPKO_00558
Lung Compartment of lung dimensionless http://purl.obolibrary.org/obo/PBPKO_00559
Arterial Compartment of arterial blood dimensionless http://purl.obolibrary.org/obo/PBPKO_00552
Venous Compartment of venous blood dimensionless http://purl.obolibrary.org/obo/PBPKO_00561
Rest Compartment of rest of the body dimensionless http://purl.obolibrary.org/obo/PBPKO_00450
Urine Compartment of urine dimensionless http://purl.obolibrary.org/obo/PBPKO_00556

Species

id name unit model qualifier
ALumen_As3 Amount of As3+ in lumen mol not specified
ALumen_As5 Amount of As5+ in lumen mol not specified
AGut_As3 Amount of As3+ in gut mol http://purl.obolibrary.org/obo/PBPKO_00496
AGut_As5 Amount of As5+ in gut mol http://purl.obolibrary.org/obo/PBPKO_00496
AGut_AsM5 Amount of MMA5 in gut mol http://purl.obolibrary.org/obo/PBPKO_00496
AGut_AsD5 Amount of DMA5 in Gut mol http://purl.obolibrary.org/obo/PBPKO_00496
AArterial_AsD5 Amount of DMA5 in arterial blood mol http://purl.obolibrary.org/obo/PBPKO_00631
ALiver_As3 Amount of As3+ in liver mol http://purl.obolibrary.org/obo/PBPKO_00497
ALiver_As5 Amount of As5+ in liver mol http://purl.obolibrary.org/obo/PBPKO_00497
ALiver_AsM3 Amount of MMA3 in liver mol http://purl.obolibrary.org/obo/PBPKO_00497
ALiver_AsM5 Amount of MMA5 in liver mol http://purl.obolibrary.org/obo/PBPKO_00497
ALiver_AsD3 Amount of DMA3 in liver mol http://purl.obolibrary.org/obo/PBPKO_00497
ALiver_AsD5 Amount od DMA5 in liver mol http://purl.obolibrary.org/obo/PBPKO_00497
ARest_As3 Amount of As3+ in rest of the body mol http://purl.obolibrary.org/obo/PBPKO_00501
ARest_As5 Amount of As5+ in rest of the body mol http://purl.obolibrary.org/obo/PBPKO_00501
ARest_AsM5 Amount of MMA5 in rest of the body mol http://purl.obolibrary.org/obo/PBPKO_00501
ARest_AsD5 Amount of DMA5 in rest of the body mol http://purl.obolibrary.org/obo/PBPKO_00501
AArterial_As3 Amount of As3+ in arterial blood mol http://purl.obolibrary.org/obo/PBPKO_00631
AArterial_As5 Amount of As5+ in arterial blood mol http://purl.obolibrary.org/obo/PBPKO_00631
AArterial_AsM5 Amount of MMA5 in arterial blood mol http://purl.obolibrary.org/obo/PBPKO_00631
AVenous_As3 Amount of As3+ in venous blood mol http://purl.obolibrary.org/obo/PBPKO_00632
AVenous_As5 Amount of As5+ in venous blood mol http://purl.obolibrary.org/obo/PBPKO_00632
AVenous_AsM5 Amount of MMA5 in venous blood mol http://purl.obolibrary.org/obo/PBPKO_00632
AVenous_AsD5 Amount of DMA5 in venous blood mol http://purl.obolibrary.org/obo/PBPKO_00632
ALung_As3 Amount of As3+ in lung mol http://purl.obolibrary.org/obo/PBPKO_00504
ALung_As5 Amount of As5+ in lung mol http://purl.obolibrary.org/obo/PBPKO_00504
ALung_AsM3 Amount of MMA3 in lung mol http://purl.obolibrary.org/obo/PBPKO_00504
ALung_AsM5 Amount of MMA5 in lung mol http://purl.obolibrary.org/obo/PBPKO_00504
ALung_AsD3 Amount of DMA3 in lung mol http://purl.obolibrary.org/obo/PBPKO_00504
ALung_AsD5 Amount of DMA5 in lung mol http://purl.obolibrary.org/obo/PBPKO_00504
AUrine_AsM3 Cumulative amount of MMA3 in urine mol http://purl.obolibrary.org/obo/PBPKO_00274
AUrine_AsD3 Cumulative amount of DMA3 in urine mol http://purl.obolibrary.org/obo/PBPKO_00274

Transfer equations

id from to equation
_J0 ALumen_As3 AGut_As3 ALumen_As3 * Ka_As3 * Frac
_J1 ALumen_As5 AGut_As5 ALumen_As5 * Ka_As5 * Frac
_J2 AGut_As3 ALiver_As3 QGut * AGut_As3 / (VGut * PG_As3)
_J3 AGut_As5 ALiver_As5 QGut * AGut_As5 / (VGut * PG_As5)
_J4 AGut_AsM5 ALiver_AsM5 QGut * AGut_AsM5 / (VGut * PG_AsM)
_J5 AGut_AsD5 ALiver_AsD5 QGut * AGut_AsD5 / (VGut * PG_AsD)
_J6 AArterial_As3 AGut_As3 QGut * AArterial_As3 / VArt
_J7 AArterial_As5 AGut_As5 QGut * AArterial_As5 / VArt
_J8 AArterial_AsM5 AGut_AsM5 QGut * AArterial_AsM5 / VArt
_J9 AArterial_AsD5 AGut_AsD5 QGut * AArterial_AsD5 / VArt
_J10 AArterial_As3 ALiver_As3 QL * AArterial_As3 / VArt
_J11 AArterial_As5 ALiver_As5 QL * AArterial_As5 / VArt
_J12 ALiver_As3 AVenous_As3 (QL + QGut) * ALiver_As3 / (VL * PL_As3)
_J13 ALiver_As5 AVenous_As5 (QL + QGut) * ALiver_As5 / (VL * PL_As5)
_J14 AArterial_AsM5 ALiver_AsM5 QL * AArterial_AsM5 / VArt
_J15 ALiver_AsM5 AVenous_AsM5 (QL + QGut) * ALiver_AsM5 / (VL * PL_AsM)
_J16 AArterial_AsD5 ALiver_AsD5 QL * AArterial_AsD5 / VArt
_J17 ALiver_AsD5 AVenous_AsD5 (QL + QGut) * ALiver_AsD5 / (VL * PL_AsD)
_J18 ALiver_As3 ALiver_As5 ALiver_As3 * kox_As3
_J19 ALiver_As5 ALiver_As3 ALiver_As5 * kred_As5
_J20 ALiver_As3 ALiver_AsM5 V_As3_MMA * ALiver_As3 / VL / ((K_As3_MMA + ALiver_As3 / VL) * (1 + ALiver_AsM3 / VL / Kinh))
_J21 ALiver_As3 ALiver_AsD5 V_As3_DMA * ALiver_As3 / VL / (K_As3_DMA + ALiver_As3 / VL)
_J22 ALiver_AsM3 ALiver_AsM5 kox_M3 * ALiver_AsM3
_J23 ALiver_AsM5 ALiver_AsM3 kred_M5 * ALiver_AsM5
_J24 ALiver_AsM3 ALiver_AsD5 V_M3_DMA * ALiver_AsM3 / VL / ((K_M3_DMA + ALiver_AsM3 / VL) * (1 + ALiver_As3 / VL / Kinh))
_J25 ALiver_AsD3 ALiver_AsD5 kox_D3 * ALiver_AsD3
_J26 ALiver_AsD5 ALiver_AsD3 kred_D5 * ALiver_AsD5
_J27 AArterial_As3 ARest_As3 QRest * AArterial_As3 / VArt
_J28 AArterial_As5 ARest_As5 QRest * AArterial_As5 / VArt
_J29 ARest_As3 AVenous_As3 QRest * ARest_As3 / (VRest * PRest_As3)
_J30 ARest_As5 AVenous_As5 QRest * ARest_As5 / (VRest * PRest_As5)
_J31 AArterial_AsM5 ARest_AsM5 QRest * AArterial_AsM5 / VArt
_J32 ARest_AsM5 AVenous_AsM5 QRest * ARest_AsM5 / (VRest * PRest_AsM)
_J33 AArterial_AsD5 ARest_AsD5 QRest * AArterial_AsD5 / VArt
_J34 ARest_AsD5 AVenous_AsD5 QRest * ARest_AsD5 / (VRest * PRest_AsD)
_J35 AVenous_As3 ALung_As3 QLung * AVenous_As3 / VVen
_J36 AVenous_As5 ALiver_As5 QLung * AVenous_As5 / VVen
_J37 ALung_As3 ALung_As5 kox_As3 * ALung_As3
_J38 ALung_As5 ALung_As3 kred_As5 * ALung_As5
_J39 ALung_As3 AArterial_As3 QLung * ALung_As3 / (VLung * PLung_As3)
_J40 ALung_As5 AArterial_As5 QLung * ALung_As5 / (VLung * PLung_As5)
_J41 AVenous_AsM5 ALung_AsM5 QLung * AVenous_AsM5 / VVen
_J42 ALung_AsM5 ALung_AsM3 kred_M5 * ALung_AsM5
_J43 ALung_AsM3 ALung_AsM5 kox_M3 * ALung_AsM3
_J44 ALung_AsM5 AArterial_AsM5 QLung * ALung_AsM5 / (VLung * PLung_AsM)
_J45 AVenous_AsD5 ALung_AsD5 QLung * AVenous_AsD5 / VVen
_J46 ALung_AsD5 ALung_AsD3 kred_D5 * ALung_AsD5
_J47 ALung_AsD3 ALung_AsD5 kox_D3 * ALung_AsD3
_J48 ALung_AsD5 AArterial_AsD5 QLung * ALung_AsD5 / (VLung * PLung_AsD)
_J49 ALiver_AsM3 AUrine_AsM3 Kurine_MMA * (ALiver_AsM3 / PL_AsM)
_J50 ALiver_AsD3 AUrine_AsD3 Kurine_DMA * (ALiver_AsD3 / PL_AsD)
_J51 ALung_AsM3 AUrine_AsM3 Kurine_MMA * ALung_AsM3 / PLung_AsM
_J52 ALung_AsD3 AUrine_AsD3 Kurine_DMA * ALung_AsD3 / PLung_AsD

ODEs

\(\frac{d[\mathtt{ALumen-As3}]}{dt} = - \mathit{ALumen_{As3}}\cdot \mathit{Ka_{As3}}\cdot \mathit{Frac}\)

\(\frac{d[\mathtt{ALumen-As5}]}{dt} = - \mathit{ALumen_{As5}}\cdot \mathit{Ka_{As5}}\cdot \mathit{Frac}\)

\(\frac{d[\mathtt{AGut-As3}]}{dt} = \mathit{ALumen_{As3}}\cdot \mathit{Ka_{As3}}\cdot \mathit{Frac} - \frac{\mathit{QGut}\cdot \mathit{AGut_{As3}}}{\mathit{VGut}\cdot \mathit{PG_{As3}}} + \frac{\mathit{QGut}\cdot \mathit{AArterial_{As3}}}{\mathit{VArt}}\)

\(\frac{d[\mathtt{AGut-As5}]}{dt} = \mathit{ALumen_{As5}}\cdot \mathit{Ka_{As5}}\cdot \mathit{Frac} - \frac{\mathit{QGut}\cdot \mathit{AGut_{As5}}}{\mathit{VGut}\cdot \mathit{PG_{As5}}} + \frac{\mathit{QGut}\cdot \mathit{AArterial_{As5}}}{\mathit{VArt}}\)

\(\frac{d[\mathtt{AGut-AsM5}]}{dt} = - \frac{\mathit{QGut}\cdot \mathit{AGut_{AsM5}}}{\mathit{VGut}\cdot \mathit{PG_{AsM}}} + \frac{\mathit{QGut}\cdot \mathit{AArterial_{AsM5}}}{\mathit{VArt}}\)

\(\frac{d[\mathtt{AGut-AsD5}]}{dt} = - \frac{\mathit{QGut}\cdot \mathit{AGut_{AsD5}}}{\mathit{VGut}\cdot \mathit{PG_{AsD}}} + \frac{\mathit{QGut}\cdot \mathit{AArterial_{AsD5}}}{\mathit{VArt}}\)

\(\frac{d[\mathtt{AArterial-AsD5}]}{dt} = - \frac{\mathit{QGut}\cdot \mathit{AArterial_{AsD5}}}{\mathit{VArt}} - \frac{\mathit{QL}\cdot \mathit{AArterial_{AsD5}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{AArterial_{AsD5}}}{\mathit{VArt}} + \frac{\mathit{QLung}\cdot \mathit{ALung_{AsD5}}}{\mathit{VLung}\cdot \mathit{PLung_{AsD}}}\)

\(\frac{d[\mathtt{ALiver-As3}]}{dt} = \frac{\mathit{QGut}\cdot \mathit{AGut_{As3}}}{\mathit{VGut}\cdot \mathit{PG_{As3}}} + \frac{\mathit{QL}\cdot \mathit{AArterial_{As3}}}{\mathit{VArt}} - \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{As3}}}{\mathit{VL}\cdot \mathit{PL_{As3}}} - \mathit{ALiver_{As3}}\cdot \mathit{kox_{As3}} + \mathit{ALiver_{As5}}\cdot \mathit{kred_{As5}} - \frac{\frac{\mathit{V\_As3\_MMA}\cdot \mathit{ALiver_{As3}}}{\mathit{VL}}}{(\mathit{K\_As3\_MMA}+\frac{\mathit{ALiver_{As3}}}{\mathit{VL}})\cdot (1+\frac{\frac{\mathit{ALiver_{AsM3}}}{\mathit{VL}}}{\mathit{Kinh}})} - \frac{\frac{\mathit{V\_As3\_DMA}\cdot \mathit{ALiver_{As3}}}{\mathit{VL}}}{\mathit{K\_As3\_DMA}+\frac{\mathit{ALiver_{As3}}}{\mathit{VL}}}\)

\(\frac{d[\mathtt{ALiver-As5}]}{dt} = \frac{\mathit{QGut}\cdot \mathit{AGut_{As5}}}{\mathit{VGut}\cdot \mathit{PG_{As5}}} + \frac{\mathit{QL}\cdot \mathit{AArterial_{As5}}}{\mathit{VArt}} - \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{As5}}}{\mathit{VL}\cdot \mathit{PL_{As5}}} + \mathit{ALiver_{As3}}\cdot \mathit{kox_{As3}} - \mathit{ALiver_{As5}}\cdot \mathit{kred_{As5}} + \frac{\mathit{QLung}\cdot \mathit{AVenous_{As5}}}{\mathit{VVen}}\)

\(\frac{d[\mathtt{ALiver-AsM3}]}{dt} = - \mathit{kox_{M3}}\cdot \mathit{ALiver_{AsM3}} + \mathit{kred_{M5}}\cdot \mathit{ALiver_{AsM5}} - \frac{\frac{\mathit{V\_M3\_DMA}\cdot \mathit{ALiver_{AsM3}}}{\mathit{VL}}}{(\mathit{K\_M3\_DMA}+\frac{\mathit{ALiver_{AsM3}}}{\mathit{VL}})\cdot (1+\frac{\frac{\mathit{ALiver_{As3}}}{\mathit{VL}}}{\mathit{Kinh}})} - \mathit{Kurine_{MMA}}\cdot \frac{\mathit{ALiver_{AsM3}}}{\mathit{PL_{AsM}}}\)

\(\frac{d[\mathtt{ALiver-AsM5}]}{dt} = \frac{\mathit{QGut}\cdot \mathit{AGut_{AsM5}}}{\mathit{VGut}\cdot \mathit{PG_{AsM}}} + \frac{\mathit{QL}\cdot \mathit{AArterial_{AsM5}}}{\mathit{VArt}} - \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{AsM5}}}{\mathit{VL}\cdot \mathit{PL_{AsM}}} + \frac{\frac{\mathit{V\_As3\_MMA}\cdot \mathit{ALiver_{As3}}}{\mathit{VL}}}{(\mathit{K\_As3\_MMA}+\frac{\mathit{ALiver_{As3}}}{\mathit{VL}})\cdot (1+\frac{\frac{\mathit{ALiver_{AsM3}}}{\mathit{VL}}}{\mathit{Kinh}})} + \mathit{kox_{M3}}\cdot \mathit{ALiver_{AsM3}} - \mathit{kred_{M5}}\cdot \mathit{ALiver_{AsM5}}\)

\(\frac{d[\mathtt{ALiver-AsD3}]}{dt} = - \mathit{kox_{D3}}\cdot \mathit{ALiver_{AsD3}} + \mathit{kred_{D5}}\cdot \mathit{ALiver_{AsD5}} - \mathit{Kurine_{DMA}}\cdot \frac{\mathit{ALiver_{AsD3}}}{\mathit{PL_{AsD}}}\)

\(\frac{d[\mathtt{ALiver-AsD5}]}{dt} = \frac{\mathit{QGut}\cdot \mathit{AGut_{AsD5}}}{\mathit{VGut}\cdot \mathit{PG_{AsD}}} + \frac{\mathit{QL}\cdot \mathit{AArterial_{AsD5}}}{\mathit{VArt}} - \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{AsD5}}}{\mathit{VL}\cdot \mathit{PL_{AsD}}} + \frac{\frac{\mathit{V\_As3\_DMA}\cdot \mathit{ALiver_{As3}}}{\mathit{VL}}}{\mathit{K\_As3\_DMA}+\frac{\mathit{ALiver_{As3}}}{\mathit{VL}}} + \frac{\frac{\mathit{V\_M3\_DMA}\cdot \mathit{ALiver_{AsM3}}}{\mathit{VL}}}{(\mathit{K\_M3\_DMA}+\frac{\mathit{ALiver_{AsM3}}}{\mathit{VL}})\cdot (1+\frac{\frac{\mathit{ALiver_{As3}}}{\mathit{VL}}}{\mathit{Kinh}})} + \mathit{kox_{D3}}\cdot \mathit{ALiver_{AsD3}} - \mathit{kred_{D5}}\cdot \mathit{ALiver_{AsD5}}\)

\(\frac{d[\mathtt{ARest-As3}]}{dt} = \frac{\mathit{QRest}\cdot \mathit{AArterial_{As3}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{ARest_{As3}}}{\mathit{VRest}\cdot \mathit{PRest_{As3}}}\)

\(\frac{d[\mathtt{ARest-As5}]}{dt} = \frac{\mathit{QRest}\cdot \mathit{AArterial_{As5}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{ARest_{As5}}}{\mathit{VRest}\cdot \mathit{PRest_{As5}}}\)

\(\frac{d[\mathtt{ARest-AsM5}]}{dt} = \frac{\mathit{QRest}\cdot \mathit{AArterial_{AsM5}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{ARest_{AsM5}}}{\mathit{VRest}\cdot \mathit{PRest_{AsM}}}\)

\(\frac{d[\mathtt{ARest-AsD5}]}{dt} = \frac{\mathit{QRest}\cdot \mathit{AArterial_{AsD5}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{ARest_{AsD5}}}{\mathit{VRest}\cdot \mathit{PRest_{AsD}}}\)

\(\frac{d[\mathtt{AArterial-As3}]}{dt} = - \frac{\mathit{QGut}\cdot \mathit{AArterial_{As3}}}{\mathit{VArt}} - \frac{\mathit{QL}\cdot \mathit{AArterial_{As3}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{AArterial_{As3}}}{\mathit{VArt}} + \frac{\mathit{QLung}\cdot \mathit{ALung_{As3}}}{\mathit{VLung}\cdot \mathit{PLung_{As3}}}\)

\(\frac{d[\mathtt{AArterial-As5}]}{dt} = - \frac{\mathit{QGut}\cdot \mathit{AArterial_{As5}}}{\mathit{VArt}} - \frac{\mathit{QL}\cdot \mathit{AArterial_{As5}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{AArterial_{As5}}}{\mathit{VArt}} + \frac{\mathit{QLung}\cdot \mathit{ALung_{As5}}}{\mathit{VLung}\cdot \mathit{PLung_{As5}}}\)

\(\frac{d[\mathtt{AArterial-AsM5}]}{dt} = - \frac{\mathit{QGut}\cdot \mathit{AArterial_{AsM5}}}{\mathit{VArt}} - \frac{\mathit{QL}\cdot \mathit{AArterial_{AsM5}}}{\mathit{VArt}} - \frac{\mathit{QRest}\cdot \mathit{AArterial_{AsM5}}}{\mathit{VArt}} + \frac{\mathit{QLung}\cdot \mathit{ALung_{AsM5}}}{\mathit{VLung}\cdot \mathit{PLung_{AsM}}}\)

\(\frac{d[\mathtt{AVenous-As3}]}{dt} = \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{As3}}}{\mathit{VL}\cdot \mathit{PL_{As3}}} + \frac{\mathit{QRest}\cdot \mathit{ARest_{As3}}}{\mathit{VRest}\cdot \mathit{PRest_{As3}}} - \frac{\mathit{QLung}\cdot \mathit{AVenous_{As3}}}{\mathit{VVen}}\)

\(\frac{d[\mathtt{AVenous-As5}]}{dt} = \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{As5}}}{\mathit{VL}\cdot \mathit{PL_{As5}}} + \frac{\mathit{QRest}\cdot \mathit{ARest_{As5}}}{\mathit{VRest}\cdot \mathit{PRest_{As5}}} - \frac{\mathit{QLung}\cdot \mathit{AVenous_{As5}}}{\mathit{VVen}}\)

\(\frac{d[\mathtt{AVenous-AsM5}]}{dt} = \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{AsM5}}}{\mathit{VL}\cdot \mathit{PL_{AsM}}} + \frac{\mathit{QRest}\cdot \mathit{ARest_{AsM5}}}{\mathit{VRest}\cdot \mathit{PRest_{AsM}}} - \frac{\mathit{QLung}\cdot \mathit{AVenous_{AsM5}}}{\mathit{VVen}}\)

\(\frac{d[\mathtt{AVenous-AsD5}]}{dt} = \frac{(\mathit{QL}+\mathit{QGut})\cdot \mathit{ALiver_{AsD5}}}{\mathit{VL}\cdot \mathit{PL_{AsD}}} + \frac{\mathit{QRest}\cdot \mathit{ARest_{AsD5}}}{\mathit{VRest}\cdot \mathit{PRest_{AsD}}} - \frac{\mathit{QLung}\cdot \mathit{AVenous_{AsD5}}}{\mathit{VVen}}\)

\(\frac{d[\mathtt{ALung-As3}]}{dt} = \frac{\mathit{QLung}\cdot \mathit{AVenous_{As3}}}{\mathit{VVen}} - \mathit{kox_{As3}}\cdot \mathit{ALung_{As3}} + \mathit{kred_{As5}}\cdot \mathit{ALung_{As5}} - \frac{\mathit{QLung}\cdot \mathit{ALung_{As3}}}{\mathit{VLung}\cdot \mathit{PLung_{As3}}}\)

\(\frac{d[\mathtt{ALung-As5}]}{dt} = \mathit{kox_{As3}}\cdot \mathit{ALung_{As3}} - \mathit{kred_{As5}}\cdot \mathit{ALung_{As5}} - \frac{\mathit{QLung}\cdot \mathit{ALung_{As5}}}{\mathit{VLung}\cdot \mathit{PLung_{As5}}}\)

\(\frac{d[\mathtt{ALung-AsM3}]}{dt} = \mathit{kred_{M5}}\cdot \mathit{ALung_{AsM5}} - \mathit{kox_{M3}}\cdot \mathit{ALung_{AsM3}} - \frac{\mathit{Kurine_{MMA}}\cdot \mathit{ALung_{AsM3}}}{\mathit{PLung_{AsM}}}\)

\(\frac{d[\mathtt{ALung-AsM5}]}{dt} = \frac{\mathit{QLung}\cdot \mathit{AVenous_{AsM5}}}{\mathit{VVen}} - \mathit{kred_{M5}}\cdot \mathit{ALung_{AsM5}} + \mathit{kox_{M3}}\cdot \mathit{ALung_{AsM3}} - \frac{\mathit{QLung}\cdot \mathit{ALung_{AsM5}}}{\mathit{VLung}\cdot \mathit{PLung_{AsM}}}\)

\(\frac{d[\mathtt{ALung-AsD3}]}{dt} = \mathit{kred_{D5}}\cdot \mathit{ALung_{AsD5}} - \mathit{kox_{D3}}\cdot \mathit{ALung_{AsD3}} - \frac{\mathit{Kurine_{DMA}}\cdot \mathit{ALung_{AsD3}}}{\mathit{PLung_{AsD}}}\)

\(\frac{d[\mathtt{ALung-AsD5}]}{dt} = \frac{\mathit{QLung}\cdot \mathit{AVenous_{AsD5}}}{\mathit{VVen}} - \mathit{kred_{D5}}\cdot \mathit{ALung_{AsD5}} + \mathit{kox_{D3}}\cdot \mathit{ALung_{AsD3}} - \frac{\mathit{QLung}\cdot \mathit{ALung_{AsD5}}}{\mathit{VLung}\cdot \mathit{PLung_{AsD}}}\)

\(\frac{d[\mathtt{AUrine-AsM3}]}{dt} = \mathit{Kurine_{MMA}}\cdot \frac{\mathit{ALiver_{AsM3}}}{\mathit{PL_{AsM}}} + \frac{\mathit{Kurine_{MMA}}\cdot \mathit{ALung_{AsM3}}}{\mathit{PLung_{AsM}}}\)

\(\frac{d[\mathtt{AUrine-AsD3}]}{dt} = \mathit{Kurine_{DMA}}\cdot \frac{\mathit{ALiver_{AsD3}}}{\mathit{PL_{AsD}}} + \frac{\mathit{Kurine_{DMA}}\cdot \mathit{ALung_{AsD3}}}{\mathit{PLung_{AsD}}}\)

Assignment rules

variable assignment
VRest BW - 0.76 - VGut - VL - VLung - VB
CLumen_As3 ALumen_As3 / Lumen
CLumen_As5 ALumen_As5 / Lumen
CGut_As3 AGut_As3 / Gut
CGut_As5 AGut_As5 / Gut
CGut_AsM5 AGut_AsM5 / Gut
CGut_AsD5 AGut_AsD5 / Gut
CLiver_As3 ALiver_As3 / Liver
CLiver_As5 ALiver_As5 / Liver
CLiver_AsM3 ALiver_AsM3 / Liver
CLiver_AsM5 ALiver_AsM5 / Liver
CLiver_AsD3 ALiver_AsD3 / Liver
CLiver_AsD5 ALiver_AsD5 / Liver
CRest_As3 ARest_As3 / Rest
CRest_As5 ARest_As5 / Rest
CRest_AsM5 ARest_AsM5 / Rest
CRest_AsD5 ARest_AsD5 / Rest
CArterial_As3 AArterial_As3 / Arterial
CArterial_As5 AArterial_As5 / Arterial
CArterial_AsM5 AArterial_AsM5 / Arterial
CArterial_AsD5 AArterial_AsD5 / Arterial
CVenous_As3 AVenous_As3 / Venous
CVenous_As5 AVenous_As5 / Venous
CVenous_AsM5 AVenous_AsM5 / Venous
CVenous_AsD5 AVenous_AsD5 / Venous
CLung_As3 ALung_As3 / Lung
CLung_As5 ALung_As5 / Lung
CLung_AsM3 ALung_AsM3 / Lung
CLung_AsM5 ALung_AsM5 / Lung
CLung_AsD3 ALung_AsD3 / Lung
CLung_AsD5 ALung_AsD5 / Lung
Ka_As3 0.004 * 60
Ka_As5 0.003 * 60
QGut 1 * 60
VArt VB / 2
QL 0.31 * 60
kred_M5 0.008 * 60
V_M3_DMA 6.6e-7 * 60
kred_D5 0.004 * 60
QRest QLung - QGut - QL
QLung 5.2 * 60
VVen VB / 2
Kurine_MMA 0.3 * 60
Kurine_DMA 0.13 * 60
Kurine_As 0.07 * 60

Initial assignments

variable assignment
Gut VGut
Liver VL
Lung VLung
Arterial VArt
Venous VVen
Rest VRest
kred_As5 0.003 * 60
V_As3_MMA 5.3e-7 * 60
V_As3_DMA 2e-6 * 60

Parameters

id name unit model qualifier
VRest Volume of rest of the body dimensionless http://purl.obolibrary.org/obo/PBPKO_00105
BW Bodyweight kg http://purl.obolibrary.org/obo/PBPKO_00008
VGut Volume of gut dimensionless http://purl.obolibrary.org/obo/PBPKO_00524
VL Volume of liver dimensionless http://purl.obolibrary.org/obo/PBPKO_00077
VLung Volume of lung dimensionless http://purl.obolibrary.org/obo/PBPKO_00097
VB Volume of blood dimensionless http://purl.obolibrary.org/obo/PBPKO_00108
CLumen_As3 Concentration of As3+ in lumen mol/L not specified
CLumen_As5 Concentration of As5+ in lumen mol/L not specified
CGut_As3 Concentration of As3+ in gut mol/L http://purl.obolibrary.org/obo/PBPKO_00538
CGut_As5 Concentration of As5+ in gut mol/L http://purl.obolibrary.org/obo/PBPKO_00538
CGut_AsM5 Concentration of MMA5 in gut mol/L http://purl.obolibrary.org/obo/PBPKO_00538
CGut_AsD5 Concentration of DMA5 in gut mol/L http://purl.obolibrary.org/obo/PBPKO_00538
CLiver_As3 Concentration of As3+ in liver mol/L http://purl.obolibrary.org/obo/PBPKO_00539
CLiver_As5 Concentration of As5+ in liver mol/L http://purl.obolibrary.org/obo/PBPKO_00539
CLiver_AsM3 Concentration of MMA3 in liver mol/L http://purl.obolibrary.org/obo/PBPKO_00539
CLiver_AsM5 Concentration of MMA5 in liver mol/L http://purl.obolibrary.org/obo/PBPKO_00539
CLiver_AsD3 Concentration of DMA3 in liver mol/L http://purl.obolibrary.org/obo/PBPKO_00539
CLiver_AsD5 Concentration of DMA5 in liver mol/L http://purl.obolibrary.org/obo/PBPKO_00539
CRest_As3 Concentration of As3+ in the rest of the body mol/L http://purl.obolibrary.org/obo/PBPKO_00548
CRest_As5 Concentration of As5+ in the rest of the body mol/L http://purl.obolibrary.org/obo/PBPKO_00548
CRest_AsM5 Concentration of MMA5 in the rest of the body mol/L http://purl.obolibrary.org/obo/PBPKO_00548
CRest_AsD5 Concentration of DMA5 in the rest of the body mol/L http://purl.obolibrary.org/obo/PBPKO_00548
CArterial_As3 Concentration of As3+ in arterial blood mol/L not specified
CArterial_As5 Concentration of As5+ in arterial blood mol/L not specified
CArterial_AsM5 Concentration of MMA5 in arterial blood mol/L not specified
CArterial_AsD5 Concentration of DMA5 in arterial blood mol/L not specified
CVenous_As3 Concentration of As3+ in venous blood mol/L not specified
CVenous_As5 Concentration of As5+ in venous blood mol/L not specified
CVenous_AsM5 Concentration of MMA5 in venous blood mol/L not specified
CVenous_AsD5 Concentration of DMA5 in venous blood mol/L not specified
CLung_As3 Concentration of As3+ in lung mol/L http://purl.obolibrary.org/obo/PBPKO_00543
CLung_As5 Concentration of As5+ in lung mol/L http://purl.obolibrary.org/obo/PBPKO_00543
CLung_AsM3 Concentration of MMA3 in lung mol/L http://purl.obolibrary.org/obo/PBPKO_00543
CLung_AsM5 Concentration of MMA5 in lung mol/L http://purl.obolibrary.org/obo/PBPKO_00543
CLung_AsD3 Concentration of DMA3 in lung mol/L http://purl.obolibrary.org/obo/PBPKO_00543
CLung_AsD5 Concentration of DMA5 in lung mol/L http://purl.obolibrary.org/obo/PBPKO_00543
Ka_As3 Oral absorption of As3+ /h http://purl.obolibrary.org/obo/PBPKO_00141
Frac Fraction of absorption dimensionless http://purl.obolibrary.org/obo/PBPKO_00263
Ka_As5 Oral absorption of As5+ /h http://purl.obolibrary.org/obo/PBPKO_00141
QGut Blood-flow to gut L/h http://purl.obolibrary.org/obo/PBPKO_00531
PG_As3 Partition coefficient Gut / Plasma of As3+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00572
PG_As5 Partition coefficient Gut / Plasma of As5+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00572
PG_AsM Partition coefficient Gut / Plasma of MMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00572
PG_AsD Partition coefficient Gut / Plasma of DMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00572
VArt Volume of arterial blood dimensionless http://purl.obolibrary.org/obo/PBPKO_00121
QL Blood-flow to liver L/h http://purl.obolibrary.org/obo/PBPKO_00024
PL_As3 Partition coefficient Liver / Plasma of As3+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00577
PL_As5 Partition coefficient Liver / Plasma of As5+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00577
PL_AsM Partition coefficient Liver / Plasma of MMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00577
PL_AsD Partition coefficient Liver / Plasma of DMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00577
kox_As3 Oxydation factor of As3+ /h not specified
kred_As5 Reduction factor of As5+ /h not specified
V_As3_MMA Maximum metabolism from As3+ to MMA mol/h http://purl.obolibrary.org/obo/PBPKO_00613
K_As3_MMA Michaelis-Menten binding constant from As3+ to MMA mol/L http://biomodels.net/SBO/SBO_0000027
Kinh Non-competitive inhibition constant mol/L http://purl.obolibrary.org/obo/PBPKO_00222
V_As3_DMA Maximum metabolism from As3+ to DMA mol/h http://purl.obolibrary.org/obo/PBPKO_00613
K_As3_DMA Michaelis-Menten binding constant from As3+ to DMA mol/L http://biomodels.net/SBO/SBO_0000027
kox_M3 Oxydation factor of MMA3 to MM5 dimensionless not specified
kred_M5 Reduction factor of MMA5 to MM3 /h not specified
V_M3_DMA Maximum metabolism from MMA3 to DMA mol/h http://purl.obolibrary.org/obo/PBPKO_00613
K_M3_DMA Michaelis-Menten binding from MMA3 to DMA mol/L http://biomodels.net/SBO/SBO_0000027
kox_D3 Oxydation factor of DMA3 to DMA5 dimensionless not specified
kred_D5 Reduction factor of DMA5 to DMA3 /h not specified
QRest Blood-flow to the rest of the body L/h http://purl.obolibrary.org/obo/PBPKO_00050
PRest_As3 Partition coefficient Restbody / Plasma of As3+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00585
PRest_As5 Partition coefficient Restbody / Plasma of As5+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00585
PRest_AsM Partition coefficient Restbody / Plasma of MMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00585
PRest_AsD Partition coefficient Restbody / Plasma of DMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00585
QLung Blood-flow to lung - Cardiac output L/h http://purl.obolibrary.org/obo/PBPKO_00013
VVen Volume of venous blood dimensionless http://purl.obolibrary.org/obo/PBPKO_00122
PLung_As3 Partition coefficient Lung / Plasma of As3+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00579
PLung_As5 Partition coefficient Lung / Plasma of As5+ dimensionless http://purl.obolibrary.org/obo/PBPKO_00579
PLung_AsM Partition coefficient Lung / Plasma of MMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00579
PLung_AsD Partition coefficient Lung / Plasma of DMA dimensionless http://purl.obolibrary.org/obo/PBPKO_00579
Kurine_MMA Urinal excretion factor of MMA /h http://purl.obolibrary.org/obo/PBPKO_00534
Kurine_DMA Urinal excretion factor of DMA /h http://purl.obolibrary.org/obo/PBPKO_00534
Age not specified y http://purl.obolibrary.org/obo/PBPKO_00521
Kurine_As Urinal excretion factor of iAs /h http://purl.obolibrary.org/obo/PBPKO_00534